Wolkenberg, Scott: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

1

Recent Progress in the Discovery of Non-Sarcosine Based GlyT1 Inhibitors

Wolkenberg, Scott, Sur, Cyrille

Journal:

Current Topics in Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 383 KB

english, 2010

2

Identification of potent agonists of photoreceptor-specific nuclear receptor (NR2E3) and preparation of a radioligand

Scott E. Wolkenberg, Zhijian Zhao, Marianna Kapitskaya, Andrea L. Webber, Konstantin Petrukhin, Yui Sing Tang, Dennis C. Dean, George D. Hartman, Craig W. Lindsley

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 133 KB

english, 2006

3

A New Method of in Situ Activation for a Novel Class of DNA Alkylating Agents: Tunable Metal Cation Complexation and Activation

Boger, Dale L., Wolkenberg, Scott E., Boyce, Christopher W.

Journal:

Journal of the American Chemical Society

Year:

2000

Language:

english

File:

PDF, 98 KB

english, 2000

4

ChemInform Abstract: Total Synthesis of Amaryllidaceae Alkaloids Utilizing Sequential Intramolecular Heterocyclic Azadiene Diels—Alder Reactions of an Unsymmetrical 1,2,4,5-Tetrazine.

Dale L. Boger, Scott E. Wolkenberg

Journal:

Year:

2001

File:

PDF, 30 KB

2001

5

DNA Alkylation Properties of Yatakemycin

Parrish, Jay P., Kastrinsky, David B., Wolkenberg, Scott E., Igarashi, Yasuhiro, Boger, Dale L.

Journal:

Journal of the American Chemical Society

Year:

2003

Language:

english

File:

PDF, 421 KB

english, 2003

6

Benzoxazolinone aryl sulfonamides as potent, selective Na v 1.7 inhibitors with in vivo efficacy in a preclinical pain model

Pero, Joseph E., Rossi, Michael A., Lehman, Hannah D.G.F., Kelly, Michael J., Mulhearn, James J., Wolkenberg, Scott E., Cato, Matthew J., Clements, Michelle K., Daley, Christopher J., Filzen, Tracey,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 425 KB

english, 2017

7

Synthesis and SAR of GlyT1 inhibitors derived from a series of N-((4-(morpholine-4-carbonyl)-1-(propylsulfonyl)piperidin-4-yl)methyl)benzamides

Zhijian Zhao, Julie A. O’Brien, Wei Lemaire, David L. Williams Jr., Marlene A. Jacobson, Cyrille Sur, Doug J. Pettibone, Philip R. Tiller, Sheri Smith, George D. Hartman, Scott E. Wolkenberg, Craig W.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 167 KB

english, 2006

8

Progress Towards Validating the NMDA Receptor Hypofunction Hypothesis of Schizophrenia

Lindsley, Craig, Shipe, William, Wolkenberg, Scott, Theberge, Cory, Williams Jr., David, Sur, Cyrille, Kinney, Gene

Journal:

Current Topics in Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 331 KB

english, 2006

9

Intramolecular Diels—Alder and Tandem Intramolecular Diels—Alder/1,3-Dipolar Cycloaddition Reactions of 1,3,4-Oxadiazoles.

Gordon D. Wilkie, Gregory I. Elliott, Brian S. J. Blagg, Scott E. Wolkenberg, Danielle R. Soenen, Michael M. Miller, Scott Pollack, Dale L. Boger

Journal:

Year:

2003

File:

PDF, 243 KB

2003

10

Reducing Limitation in Probe Design: The Development of a Diazirine-Compatible Suzuki–Miyaura Cross Coupling Reaction

Ichiishi, Naoko, Moore, Keith P., Wassermann, Anne Mai, Wolkenberg, Scott E., Krska, Shane W.

Journal:

ACS Medicinal Chemistry Letters

Year:

2018

Language:

english

File:

PDF, 1.65 MB

english, 2018

11

Mechanisms of in situ Activation for DNA-Targeting Antitumor Agents

Scott E. Wolkenberg, Dale L. Boger

Journal:

Year:

2002

File:

PDF, 24 KB

2002

12

Discovery of ethyl ketone-based HDACs 1, 2, and 3 selective inhibitors for HIV latency reactivation

Yu, Wensheng, Liu, Jian, Yu, Younong, Zhang, Vivian, Clausen, Dane, Kelly, Joseph, Wolkenberg, Scott, Beshore, Douglas, Duffy, Joseph L., Chung, Christine C., Myers, Robert W., Klein, Daniel J., Fells

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.25 MB

2020

13

Controlled derivatization of polyhalogenated quinolines utilizing selective cross-coupling reactions

M. Brad Nolt, Zhijian Zhao, Scott E. Wolkenberg

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 125 KB

english, 2008

14

Discovery of GlyT1 inhibitors with improved pharmacokinetic properties

Scott E. Wolkenberg, Zhijian Zhao, David D. Wisnoski, William H. Leister, Julie O’Brien, Wei Lemaire, David L. Williams Jr., Marlene A. Jacobson, Cyrille Sur, Gene G. Kinney, Doug J. Pettibone, Philip

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 1.24 MB

english, 2009

15

Synthesis and Evaluation of 1,2,8,8a-Tetrahydrocyclopropa[ c ]pyrrolo[3,2- e ]indol-4(5 H )-one, the Parent Alkylation Subunit of CC-1065 and the Duocarmycins: Impact of the Alkylation Subunit Substituents and Its Implications for DNA Alkylation Catalysis

Boger, Dale L., Santillán, Alejandro, Searcey, Mark, Brunette, Steven R., Wolkenberg, Scott E., Hedrick, Michael P., Jin, Qing

Journal:

Journal of Organic Chemistry

Year:

2000

Language:

english

File:

PDF, 356 KB

english, 2000

16

Rational Design, Synthesis, and Evaluation of Key Analogues of CC-1065 and the Duocarmycins

Tichenor, Mark S., MacMillan, Karen S., Stover, James S., Wolkenberg, Scott E., Pavani, Maria G., Zanella, Lorenzo, Zaid, Abdel N., Spalluto, Gianpiero, Rayl, Thomas J., Hwang, Inkyu, Baraldi, Pier Gi

Journal:

Journal of the American Chemical Society

Year:

2007

Language:

english

File:

PDF, 718 KB

english, 2007

17

In vitro Characterization of MK-3328: A Novel Fluorinated Positron Emission Tomography Tracer for Plaques

Cyrille Sur, Zhizhen Zeng, Eric Hostetler, Brett M. Connolly, Patricia J. Miller, Stacey O'Malley, Tsin-Bau Chen, Christopher Culberson, Scott Harrison, Jim Mulhearn, Scott Wolkenberg, James Barrow, S

Journal:

Alzheimer's & Dementia

Year:

2010

Language:

english

File:

PDF, 49 KB

english, 2010

18

Combinatorial Synthesis and Discovery of an Antibiotic Compound. An Experiment Suitable for High School and Undergraduate Laboratories

Wolkenberg, Scott E., Su, Andrew I.

Journal:

Journal of Chemical Education

Year:

2001

Language:

english

File:

PDF, 77 KB

english, 2001

19

Total Synthesis and Evaluation of Cytostatin, Its C10−C11 Diastereomers, and Additional Key Analogues: Impact on PP2A Inhibition

Lawhorn, Brian G., Boga, Sobhana B., Wolkenberg, Scott E., Colby, David A., Gauss, Carla-Maria, Swingle, Mark R., Amable, Lauren, Honkanen, Richard E., Boger, Dale L.

Journal:

Journal of the American Chemical Society

Year:

2006

Language:

english

File:

PDF, 793 KB

english, 2006

20

General Microwave-Assisted Protocols for the Expedient Synthesis of Quinoxalines and Heterocyclic Pyrazines.

Zhijian Zhao, David D. Wisnoski, Scott E. Wolkenberg, William H. Leister, Yi Wang, Craig W. Lindsley

Journal:

Year:

2004

File:

PDF, 36 KB

2004

21

[18F]Fluoroazabenzoxazoles as potential amyloid plaque PET tracers: synthesis and in vivo evaluation in rhesus monkey

Eric D. Hostetler, Sandra Sanabria-Bohórquez, Hong Fan, Zhizhen Zeng, Linda Gammage, Patricia Miller, Stacey O'Malley, Brett Connolly, James Mulhearn, Scott T. Harrison, Scott E. Wolkenberg, James C.

Journal:

Nuclear Medicine and Biology

Year:

2011

Language:

english

File:

PDF, 846 KB

english, 2011

22

Intramolecular Diels−Alder and Tandem Intramolecular Diels−Alder/1,3-Dipolar Cycloaddition Reactions of 1,3,4-Oxadiazoles

Wilkie, Gordon D., Elliott, Gregory I., Blagg, Brian S. J., Wolkenberg, Scott E., Soenen, Danielle R., Miller, Michael M., Pollack, Scott, Boger, Dale L.

Journal:

Journal of the American Chemical Society

Year:

2002

Language:

english

File:

PDF, 147 KB

english, 2002

23

Progress in the Preparation and Testing of Glycine Transporter Type-1 (GlyT1) Inhibitors

Lindsley, Craig, Wolkenberg, Scott, Kinney, Gene

Journal:

Current Topics in Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 91 KB

english, 2006

24

Accelerating lead development by microwave-enhanced medicinal chemistry

William D. Shipe, Scott E. Wolkenberg, Craig W. Lindsley

Journal:

Drug Discovery Today: Technologies

Year:

2005

Language:

english

File:

PDF, 183 KB

english, 2005

25

Efficient Synthesis of Imidazoles from Aldehydes and 1,2-Diketones Using Microwave Irradiation.

Scott E. Wolkenberg, David D. Wisnoski, William H. Leister, Yi Wang, Zhijian Zhao, Craig W. Lindsley

Journal:

Year:

2004

File:

PDF, 140 KB

2004

26

The synthesis and preclinical evaluation in rhesus monkey of [18F]MK-6577 and [11C]CMPyPB glycine transporter 1 positron emission tomography radiotracers

Terence G. Hamill, Waisi Eng, Andrew Jennings, Richard Lewis, Steven Thomas, Suzanne Wood, Leslie Street, David Wisnoski, Scott Wolkenberg, Craig Lindsley, Sandra M. Sanabria-BohÓRquez, Shil Patel, Ke

Journal:

Year:

2011

Language:

english

File:

PDF, 1.36 MB

english, 2011

27

Synthesis and Evaluation of 5-Fluoro-2-aryloxazolo[5,4- b ]pyridines as β-Amyloid PET Ligands and Identification of MK-3328

Harrison, Scott T., Mulhearn, James, Wolkenberg, Scott E., Miller, Patricia J., O’Malley, Stacey S., Zeng, Zhizhen, Williams, David L., Hostetler, Eric D., Sanabria-Bohórquez, Sandra, Gammage, Linda,

Journal:

ACS Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 3.23 MB

english, 2011

28

Design, Synthesis, and Evaluation of Novel 3,6-Diaryl-4-aminoalkoxyquinolines as Selective Agonists of Somatostatin Receptor Subtype 2

Wolkenberg, Scott E., Zhao, Zhijian, Thut, Catherine, Maxwell, Jill W., McDonald, Terrence P., Kinose, Fumi, Reilly, Michael, Lindsley, Craig W., Hartman, George D.

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 1.42 MB

english, 2011

29

Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs)

Zhijian Zhao, Scott E. Wolkenberg, Meiqing Lu, Vandna Munshi, Gregory Moyer, Meizhen Feng, Anthony V. Carella, Linda T. Ecto, Lori J. Gabryelski, Ming-Tain Lai, Sridar G. Prasad, Youwei Yan, Georgia B

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 272 KB

english, 2008

30

Corrigendum to “Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs)” [Bioorg. Med. Chem. Lett. (2008) 554]

Zhijian Zhao, Scott E. Wolkenberg, Philip E.J. Sanderson, Meiqing Lu, Vandna Munshi, Gregory Moyer, Meizhen Feng, Anthony V. Carella, Linda T. Ecto, Lori J. Gabryelski, Ming-Tain Lai, Sridar G. Prasad

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 109 KB

english, 2010

31

Total Synthesis of Anhydrolycorinone Utilizing Sequential Intramolecular Diels−Alder Reactions of a 1,3,4-Oxadiazole

Wolkenberg, Scott E., Boger, Dale L.

Journal:

Journal of Organic Chemistry

Year:

2002

Language:

english

File:

PDF, 91 KB

english, 2002

32

Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics

Wolkenberg, Scott E., Nolt, M. Brad, Bilodeau, Mark T., Trotter, B. Wesley, Manley, Peter J., Kett, Nathan R., Nanda, Kausik K., Wu, Zhicai, Cato, Matthew J., Kane, Stefanie A., Kiss, Laszlo, Spencer,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 1.21 MB

english, 2017

33

General microwave-assisted protocols for the expedient synthesis of quinoxalines and heterocyclic pyrazines

Zhijian Zhao, David D Wisnoski, Scott E Wolkenberg, William H Leister, Yi Wang, Craig W Lindsley

Journal:

Tetrahedron Letters

Year:

2004

Language:

english

File:

PDF, 312 KB

english, 2004

34

Total Synthesis of Amaryllidaceae Alkaloids Utilizing Sequential Intramolecular Heterocyclic Azadiene Diels−Alder Reactions of an Unsymmetrical 1,2,4,5-Tetrazine

Boger, Dale L., Wolkenberg, Scott E.

Journal:

Journal of Organic Chemistry

Year:

2000

Language:

english

File:

PDF, 78 KB

english, 2000

35

Characterization of Non-Nitrocatechol Pan and Isoform Specific Catechol- O -methyltransferase Inhibitors and Substrates

Robinson, Ronald G., Smith, Sean M., Wolkenberg, Scott E., Kandebo, Monika, Yao, Lihang, Gibson, Christopher R., Harrison, Scott T., Polsky-Fisher, Stacey, Barrow, James C., Manley, Peter J., Mulhearn

Journal:

ACS Chemical Neuroscience

Year:

2012

Language:

english

File:

PDF, 1.72 MB

english, 2012

36

Metal Cation Complexation and Activation of Reversed CPyI Analogues of CC-1065 and Duocarmycin SA: Partitioning the Effects of Binding and Catalysis

Ellis, David A., Wolkenberg, Scott E., Boger, Dale L.

Journal:

Journal of the American Chemical Society

Year:

2001

Language:

english

File:

PDF, 215 KB

english, 2001

37

High concentration electrophysiology-based fragment screen: Discovery of novel acid-sensing ion channel 3 (ASIC3) inhibitors

Scott E. Wolkenberg, Zhijian Zhao, James J. Mulhearn, Scott T. Harrison, John M. Sanders, Matthew J. Cato, Aneta Jovanovska, Jacqueline Panigel, Sean P. Cook, Darrell A. Henze, Stefanie A. Kane, Georg

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 985 KB

english, 2011

38

Efficient Synthesis of Imidazoles from Aldehydes and 1,2-Diketones Using Microwave Irradiation

Wolkenberg, Scott E., Wisnoski, David D., Leister, William H., Wang, Yi, Zhao, Zhijian, Lindsley, Craig W.

Journal:

Organic Letters

Year:

2004

Language:

english

File:

PDF, 66 KB

english, 2004

39

Convenient and General Microwave-Assisted Protocols for the Expedient Synthesis of Heterocycles

D. Shipe, William, Yang, Feng, Zhao, Zhijian, E. Wolkenberg, Scott, Brad Nolt, M., W. Lindsley, Craig

Journal:

Year:

2006

Language:

english

File:

PDF, 397 KB

english, 2006

40

Mechanisms of in Situ Activation for DNA-Targeting Antitumor Agents

Wolkenberg, Scott E., Boger, Dale L.

Journal:

Chemical Reviews

Year:

2002

Language:

english

File:

PDF, 320 KB

english, 2002

41

Convenient preparation of substituted 5-aminooxazoles via a microwave-assisted Cornforth rearrangement

M. Brad Nolt, Mark A. Smiley, Sandor L. Varga, Ray T. McClain, Scott E. Wolkenberg, Craig W. Lindsley

Journal:

Year:

2006

Language:

english

File:

PDF, 391 KB

english, 2006

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски